Inhibition of the subgenomic hepatitis C virus replicon in huh-7 cells by 2'-deoxy-2'-fluorocytidine.

نویسندگان

  • Lieven J Stuyver
  • Tamara R McBrayer
  • Tony Whitaker
  • Phillip M Tharnish
  • Mangala Ramesh
  • Stefania Lostia
  • Leanne Cartee
  • Junxing Shi
  • Ann Hobbs
  • Raymond F Schinazi
  • Kyoichi A Watanabe
  • Michael J Otto
چکیده

2'-Deoxy-2'-fluorocytidine (FdC) is a potent inhibitor of the hepatitis C virus RNA replicon in culture, and FdC-5'-triphosphate is an effective inhibitor of the NS5B polymerase. Dynamic profiling of cell growth in an antiviral assay showed that FdC caused cytostasis due to an S-phase arrest. These observations demonstrate that FdC treatment is affecting both a viral target and a cellular target.

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عنوان ژورنال:
  • Antimicrobial agents and chemotherapy

دوره 48 2  شماره 

صفحات  -

تاریخ انتشار 2004